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Product name : CP-673451
Item : cc529
Price : 10mg, $275; 50mg, $895; 100mg, $1295; 200mg, $2095
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
Additional Information : We offer significant discount for bulky quantity order
CAS : 
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Details:
CP-673451 is a potent inhibitor of platelet-derived growthfactor ß-receptor (PDGFR-ß) kinase- andPDGF-BB-stimulated autophosphorylation of PDGFR-ßin cells (IC50 = 1 nmol/L) being more than 450-fold selectivefor PDGFR-ß versus other angiogenic receptors (e.g.,vascular endothelial growth factor receptor 2, TIE-2, and fibroblastgrowth factor receptor 2). CP 673451 did not inhibit vascular endothelial growth factor- or basic fibroblast growth factor-induced angiogenesis at concentrations which inhibited tumor growth. [1]
                                                                                                                
Reference:
[1] Cancer Res. 2005, 65, 957-966.
 
 
Chemical Information
Molecular Weight (WM):
417.50
Formula:
C24H27N5O2
CAS No:
343787-29-1
Purity:
≥ 98%
Synonyms:
CP673451
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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