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Product name : Saxagliptin (BMS 477118)
Item : cc226
Price : 200mg, $459;500mg, $850; 1g $1195; 2g, $1795
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 361442-04-8
Molecular Weight : 315.41
Formula : C₁₈H₂₅N₃O₂
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
Saxagliptin (BMS-477118), is a new oral hypoglycemic (anti-diabetic drug) of the new dipeptidyl peptidase-4 (DPP-4) inhibitor with IC50 of 50 nM. It increases the circulating levels of incretin hormones (GLP-1, GIP), which contributes to amplify the insulin secretory response to meals and to reduce postprandial hyperglycaemia and, subsequently, fasting glycaemia.   [1][2]
 
Reference:
[1] J Pharmacol. Pharmacother. 2011, 2, 230-235.
[2] Rev. Med. Liege 2010, 65, 527-532.
 
 
Chemical Information
Molecular Weight (WM):
315.41
Formula:
C18H25N3O2
CAS No:
361442-04-8
Purity:
≥ 98%
Synonyms:
Onglyza, BMS477118
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.
 
 

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