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Product name : Anacetrapib (MK 0859)
Item : cc77
Price : 10mg, $295; 50mg, $795; 100mg, $1395; 200mg, $2395
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
Additional Information : We offer significant discount for bulky quantity order
CAS : 
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Details:
Anacetrapib (MK-0859) is a potent and selective rhCETP and C13S CETP mutant inhibitor with IC50 of 7.9 nM and 11.8 nM, respectively. Anacetrapib (MK0859) is not only able to increase HDL-cholesterol, but also further decreases LDL-cholesterol when taken in combination with a statin. Anacetrapib dose-dependently and significantly decreases the transfer of CE from HDL3 to HDL2.   [1][2]
 
Reference:
[1] J Lipid Res. 2010, 51, 3443-3454.
[2] Drug Metab. Dispos. 2010, 38, 459-473.
 
 
Chemical Information
Molecular Weight (WM):
637.51
Formula:
C30H25F10NO3
CAS No:
875446-37-0
Purity:
≥ 98%
Synonyms:
MK 0859
 
DMSO ≥ 127 mg/mL
Solubility (25℃)
Water < 1 mg/mL
 
Ethanol ≥ 127 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.
 

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