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Product name : Sitagliptin (MK 0431)
Item : cc318
Price : 200mg, $55; 500mg, $125; 1g, $195
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
Additional Information : We offer significant discount for bulky quantity order
CAS : 
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Details:
Sitagliptin phosphate (MK-0431) is a potent, orally active inhibitor of DPP-IV with an IC50 of 19 nM in Caco-2 cell extracts. [1][2]
 
Reference:
[1] J Pharmacol. Exp. Ther. 2008, 325, 175-182.
[2] Diabetes 2009, 58, 641-651.
 
 
Chemical Information
Molecular Weight (WM):
523.32
Formula:
C16H15F6N5O.H3PO4.H2O
CAS No:
654671-77-9, 486460-32-6 (free base), 654671-78-0 (phosphate)
Purity:
≥ 98%
Synonyms:
MK0431
 
DMSO ≥ 101 mg/mL
Solubility (25℃)
Water ≥ 101 mg/mL
 
Ethanol < 1 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.
 

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