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Product name : GSK 256066
Item : cc33
Price : 200mg, $1250;500mg, $2090; 1g $2995; 2g, $4395
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 801312-28-7
Molecular Weight : 518.58
Formula : C₂₇H₂₆N₄O₅S
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
GSK256066 is a selective PED4B inhibitor with IC50 of 3.2 pM. GSK-256066 has been demonstrated to have exceptional potency in vitro and in vivo and is being clinically investigated as a treatment for chronic obstructive pulmonary disease.  [1][2]
 
Reference:
[1] J Pharmacol. Exp. Ther. 2011, 337, 145-154.
[2] Bioorg. Med. Chem. Lett. 2009, 19, 5261-5265.
 

Chemical Information
Molecular Weight (WM):
518.58
Formula:
C27H26N4O5S
CAS No:
801312-28-7, 801311-47-7 (XHCl), 801315-14-0 (HCl)
Purity:
≥ 98%
Synonyms:
GSK 256066
 
DMSO ≥ 5 mg/mL
Solubility (25℃)
Water < 1 mg/mL
 
Ethanol < 1 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.
 

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