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Products > GPCR > Endothelin Receptor > sitaxsentan(TBC 11251)
Product name : sitaxsentan(TBC 11251)
Item : cc390
Price : 200mg, $1250;500mg, $2090; 1g $2995; 2g, $4395
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 184036-34-8
Molecular Weight : 454.9
Formula : C₁₈H₁₅ClN₂O₆S₂
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
Sitaxentan (TBC-11251) is a small molecule that blocks the action of endothelin (ET) on the endothelin-A (ETA) receptor selectively (by a factor of 6000 compared to the ETB). [1][2]
 
Reference:
[1] Ann. Rheum. Dis. 2007, 66, 1467-1472.
[2] Int. J Cardiol. 2010, 144, e43-45.
 
 
Chemical Information
Molecular Weight (WM):
454.91
Formula:
C18H15ClN2O6S2
CAS No:
184036-34-8, 210421-64-0 (sodiem salt)
Purity:
≥ 98%
Synonyms:
TBC 11251
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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