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Product name : AS 604850
Item : cc611
Price : 200mg, $1250;500mg, $2090; 1g $2995; 2g, $4395
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 648449-76-7
Molecular Weight : 285.22
Formula : C11H5F2NO4S
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
AS-604850 is a selective, ATP-competitive PI3Kγ inhibitor with IC50 of 250 nM. AS604850 is ATP-competitive PI3Kγ inhibitor with Ki values of 0.18 μM. AS 604850 is isoform selective inhibitor of PI3Kγ with over 30-fold selectivity for PI3Kγ and β, and 18-fold selectivity over PI3Kα. (PI3Kα: IC50 = 4.5 μM, PI3Kγ and β: IC50 > 20μM).  [1][2]
 
Reference:
[1] J Hepatol. 2010, 53, 918-925.
[2] Nat. Med. 2005, 11, 936-943.
 
 
Chemical Information
Molecular Weight (WM):
285.22
Formula:
C11H5F2NO4S
CAS No:
648449-76-7
Purity:
≥ 98%
Synonyms:
 
 
DMSO ≥ 57 mg/mL
Solubility (25℃)
Water < 1 mg/mL
 
Ethanol ≥ 5 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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