Product name : MK 3207
Item : cc623
Price : 200mg, $1750;500mg, $2690; 1g $3590; 2g, $5190
contact : Send enquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 957118-49-9
Molecular Weight : 557.59
Formula : C₃₁H₂₉F₂N₅O₃
Storage : at -20°C
Additional information : We offer significant discount for larger quantity order
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MK-3207 is a calcitonin gene-related peptide (CGRP) receptor antagonist with IC50 of 0.12 nM. MK3207 displays marked selectivity for human CGRP receptor versus related human AM1 (CLR/RAMP2) receptor, AM2 (CLR/RAMP3) receptor, AMY3 (CTR/RAMP3) receptor, and CTR with Ki values of 16.5 μM, 0.156 μM, 0.128 μM and 1.9 μM, respectively. [1][2]
Reference:
[1] J Pharmacol. Exp. Ther. 2010, 333, 152-160.
[2] ACS Med. Chem. Lett. 2010, 1, 24-29.
Chemical Information
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE. |
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