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Product name : Tariquidar (XR 9576)
Item : cc775
Price : 200mg, $750;500mg, $1290; 1g, $1990; 2g, $2995
contact : Send inquiry to: info@acesobio.com
CAS : 206873-63-4
Molecular Weight : 646.73
Formula : C₃₈H₃₈N₄O₆
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
Tariquidar (XR-9576) is a P-glycoprotein inhibitor undergoing research as an adjuvant against multidrug resistance in cancer. Tariquidar non-competitively binds to the p-glycoprotein transporter, thereby inhibiting transmembrane transport of anticancer drugs. Inhibition of transmembrane transport may result in increased intracellular concentrations of an anticancer drug, thereby augmenting its cytotoxicity. [1][2]
 
Reference:
[1] J Med. Chem. 2011, 54, 5878-5889.
[2] J Biol. Chem. 2012, 287, 26806-20816.
 
Chemical Information
Molecular Weight (WM):
646.73
Formula:
C38H38N4O6
CAS No:
206873-63-4
Purity:
≥ 98%
Synonyms:
XR9576
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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