Favorite  |  Set Home
Products > PARP > > Inolitazone (Efatutazone)
Product name : Inolitazone (Efatutazone)
Item : cc782
Price : 5mg, $375; 10mg, $595; 50mg, $2795;
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239
Additional Information : We offer significant discount for bulky quantity order
CAS : 
 Enlarge Image                   Back
             [Next Product]→


Details:
Inolitazone (Efatutazone) is an orally bioavailable PAPR-gamma inhibitor with potential antineoplastic activity. Inolitazone binds to and activates peroxisome proliferation-activated receptor gamma (PPAR-gamma), which may result in the induction of tumor cell differentiation and apoptosis, and so a reduction in tumor cell proliferation. PPAR-gamma is a nuclear hormone receptor and ligand-activated transcription factor controlling gene expression involved in such cellular processes as differentiation, apoptosis, cell-cycle control, carcinogenesis, and inflammation. [1][2]
 
Reference:
[1] Biochem. J 2005, 389 (Pt 3) 913-918.
[2] J Pharmacol. Exp. Ther. 2005, 312, 1027-1033.
 
Chemical Information
Molecular Weight (WM):
502.58
Formula:
C27H26N4O4S
CAS No:
223132-37-4
Purity:
≥ 98%
Synonyms:
CS-7017, RS5444
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

Related Products :
Iniparib (BSI-201)
Iniparib (BSI-201)
Price: 10mg, $110; 50mg, $295; 100mg, $575; 200mg, $895
Olaparib (AZD2281)
Olaparib (AZD2281)
Price: 10mg, $60; 50mg, $195; 100mg, $295; 200mg; $495
ABT 888 (Veliparib)
ABT 888 (Veliparib)
Price: 10mg, $110; 50mg, $295; 100mg, $475; 200mg, $895
Rucaparib (AG 014699, PF 01367338)
Rucaparib (AG 014699, PF 01367338)
Price: 10mg, $140; 50mg,$595; 100mg, $895; 200mg,$1895
AG 14361
AG 14361
Price: 10mg, $295; 50mg, $955; 100mg, $1295; 200mg, $1995
Atopaxar (E 5555)
Atopaxar (E 5555)
Price: 10mg, $375; 50mg, $975; 100mg, $1495;200mg, $2295