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Product name : Inolitazone (Efatutazone)
Item : cc782
Price : 200mg, $950;500mg, $1695; 1g, $2490; 2g, $3590
contact : Send inquiry to: info@acesobio.com
CAS : 223132-37-4
Molecular Weight : 502.58
Formula : C₂₇H₂₆N₄O₄S
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
Inolitazone (Efatutazone) is an orally bioavailable PAPR-gamma inhibitor with potential antineoplastic activity. Inolitazone binds to and activates peroxisome proliferation-activated receptor gamma (PPAR-gamma), which may result in the induction of tumor cell differentiation and apoptosis, and so a reduction in tumor cell proliferation. PPAR-gamma is a nuclear hormone receptor and ligand-activated transcription factor controlling gene expression involved in such cellular processes as differentiation, apoptosis, cell-cycle control, carcinogenesis, and inflammation. [1][2]
 
Reference:
[1] Biochem. J 2005, 389 (Pt 3) 913-918.
[2] J Pharmacol. Exp. Ther. 2005, 312, 1027-1033.
 
Chemical Information
Molecular Weight (WM):
502.58
Formula:
C27H26N4O4S
CAS No:
223132-37-4
Purity:
≥ 98%
Synonyms:
CS-7017, RS5444
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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