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Products > Cell Metabolism > DPP4 > Trelagliptin(SYR-472)
Product name : Trelagliptin(SYR-472)
Item : CR1863
Price : 1g, $650;2g, $1050;
contact : Send inquiry to: info@acesobio.com
CAS : 1029877-94-8
Molecular Weight : 475.47
Formula : C₂₂H₂₆FN₅O₆
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
 Chemical Information
M.Wt 475.47 Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Formula C22H26FN5O6
CAS No 1029877-94-8
Solubility

DMSO

Biological Activity of Trelagliptin succinate

 

Trelagliptin(SYR-472) is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D).
IC50 value:
Target: DPP4
Two Phase II clinical studies have been completed with Efficacy and Safety of SYR-472 in Subjects With Type 2 Diabetes Mellitus. Phase III clinical studies with trelagliptin in Japan to evaluate its safety and efficacy in a once-weekly oral treatment regimen. Currently, all available DPP-4 inhibitors are dosed once-daily. A once-weekly treatment, such as trelagliptin, would provide patients with a convenient treatment alternative and has the potential to improve treatment compliance.

 

Clinical Information of Trelagliptin succinate

MORE

[1]. Efficacy of SYR-472 in Subjects With Type 2 Diabetes Mellitus

[2]. Efficacy and Safety of SYR-472 in Subjects With Type 2 Diabetes Mellitus

[3]. Long-term Study of SYR-472

[4]. SYR-472 Open-label Study

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