Favorite  |  Set Home
Products > Others > > Rolapitant
Product name : Rolapitant
Item : CR1837
Price : 100mg, $845; 200mg, $1285
contact : Send inquiry to: info@acesobio.com
Additional Information :  We offer significant discount for bulky quantity order,Please ask price and availability of other quantities
CAS : 552292-08-7
 Enlarge Image                   Back
←[Previous Product]              [Next Product]→


Details:
 Name: Rolapitant

CAS# 552292-08-7

Chemical Formula: C25H26F6N2O2

Exact Mass: 500.18985

Molecular Weight: 500.48

Elemental Analysis: C, 60.00; H, 5.24; F, 22.78; N, 5.60; O, 6.39


Description of rolapitant: Rolapitant, also known as SCH-619734, is a selective, bioavailable, CNS penetrant neurokinin NK1 receptor antagonist that shows behavioral effects in animals models of emesis. In vitro studies indicate that rolapitant has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold. Rolapitant is a functionally competitive antagonist, as measured by calcium efflux, with a calculated Kb of 0.17 nM.



Related Products :
Netobimin
Netobimin
Price: 10mg, $125; 50mg, $495; 100mg, $695; 200mg, $1095
Aprepitant (MK 0869)
Aprepitant (MK 0869)
Price: 10mg, $295; 50mg, $895; 100mg, $1295; 200mg, $1995
BMS 309403
BMS 309403
Price: 10mg, $295; 50mg, $995; 100mg,$1495; 200mg, $2295
QS 11
QS 11
Price: 10mg, $95, 50mg, $375; 100mg, $655; 200mg, $1295
GIT 27
GIT 27
Price: 200mg, $845; 500mg, $1285
P005672
P005672
Price: 10mg, $195; 50mg, $595; 100mg, $995; 200mg, $1695
Plerixafor (DB 06809, Mozobil, AMD 3100)
Plerixafor (DB 06809, Mozobil, AMD 3100)
Price: 10mg, $95, 50mg, $295; 100mg, $475; 200mg, $695
P7C3
P7C3
Price: 100mg, $745; 200mg, $1185