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Product name : Rolapitant
Item : CR1837
Price : 200mg, $950;500mg, $1695; 1g, $2490; 2g, $3590
contact : Send inquiry to: info@acesobio.com
CAS : 552292-08-7
Molecular Weight : 500.48
Formula : C₂₅H₂₆F₆N₂O₂
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
 Name: Rolapitant

CAS# 552292-08-7

Chemical Formula: C25H26F6N2O2

Exact Mass: 500.18985

Molecular Weight: 500.48

Elemental Analysis: C, 60.00; H, 5.24; F, 22.78; N, 5.60; O, 6.39


Description of rolapitant: Rolapitant, also known as SCH-619734, is a selective, bioavailable, CNS penetrant neurokinin NK1 receptor antagonist that shows behavioral effects in animals models of emesis. In vitro studies indicate that rolapitant has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold. Rolapitant is a functionally competitive antagonist, as measured by calcium efflux, with a calculated Kb of 0.17 nM.



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