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Product name : Enzalutamide (MDV3100)
Item : cc-412
Price : 5g, $650;10g, $1050; 20g $1650
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 915087-33-1
Molecular Weight : 464.44
Formula : C₂₁H₁₆F₄N₄O₂S
Storage : at -20°C
Additional information : We offer significant discount for larger quantity order
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Details:
Enzalutamide (MDV3100) is an experimental androgen receptor antagonist drug developed by the pharmaceutical company Medivation for the treatment of castration-resistant prostate cancer currently in phase 3 clinical trials. Results so far have been encouraging; Medivation has reported up to an 89% decrease in prostate specific antigen serum levels after a month of taking the medicine. Early preclinical studies also suggest that enzalutamide inhibits breast cancer cell growth.[1][2]
 
Reference:
[1] Science 2009, 324, 787-790.
[2] J Med. Chem. 2010, 53, 2779-2796.
 
 
Chemical Information
Molecular Weight (WM):
464.44
Formula:
C21H16F4N4O2S
CAS No:
915087-33-1
Purity:
≥ 98%
Synonyms:
MDV-3100, MDV 3100
 
DMSO ≥ 93 mg/mL
Solubility: (R.T.: 25℃):
Water < 1 mg/mL
 
Ethanol ≥ 17 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.
 
 

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