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Product name : Iniparib (BSI-201)
Item : cc-485
Price : 10mg, $110; 50mg, $295; 100mg, $575; 200mg, $895
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
Additional Information : We offer significant discount for larger quantity order
CAS : 
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Details:
Iniparib (BSI-201) is a potent PARP1 inhibitor with strong anti-neoplastic effect. BSI-201 covalently binds and inhibits PARP-1. When given as a single agent and in combination with other cytotoxic agents, Iniparib (BSI-201) is active against a broad range of cancer cells in culture.Iniparib (BSI-201) has first-in-class and best-in-class potential as targeted therapy for several types of cancer. Iniparib (BSI-201) has demonstrated activity in multiple types of solid tumors, with prolonged inhibition of its target. Iniparib (BSI-201) has shown a strong safety profile. Iniparib (BSI-201) is a leading candidate in the field of PARP inhibitors and is the furthest along in clinical development of this novel therapeutic approach. [1][2]
 
Reference:
[1] Clin. Cancer Res. 2012, 18, 510-523.
[2] Clin. Cancer Res. 2012, 18, 1655-1662.
 
 
Chemical Information
Molecular Weight (WM):
292.03
Formula:
C7H5IN2O3
CAS No:
160003-66-7
Purity:
≥ 98%
Synonyms:
BSI 201, NSC 746045, IND 71677, BSI201
 
DMSO ≥ 58 mg/mL
Solubility: (R.T.: 25℃):
Water < 1 mg/mL
 
Ethanol ≥ 37 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.
 
 

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