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Product name : Dapagliflozin (BMS 512148)
Item : cc205
Price : 10mg, $275; 50mg, $795; 100mg, $1295; 200mg, $1995
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
Additional Information : We offer significant discount for bulky quantity order
CAS : 
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Details:
Dapagliflozin (BMS-512148) is a potent and selective sodium-glucose transport proteins (SGLT2) inhibitor with EC50 of 1.1 nM. SGLT2 is responsible for at least 90% of the glucose reabsorption in the kidney. Blocking this transporter causes blood glucose to be eliminated through the urine. [1][2]
 
Reference:
[1] Diabetes Obes. Metab. 2010, 12, 1004-1012.
[2] J Med. Chem. 2008, 51, 1145-1149.
 
 
Chemical Information
Molecular Weight (WM):
408.87
Formula:
C21H25ClO6
CAS No:
461432-26-8, 960404-48-2 ((2S)-1,2-propanediol, hydrate)
Purity:
≥ 98%
Synonyms:
BMS512148 BMS 512148
 
DMSO ≥ 82 mg/mL
Solubility (25℃)
Water < 1 mg/mL
 
Ethanol ≥ 82 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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