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GSK 126
GSK-126 is a potent, highly selective, S-adenosyl-methionine-competitive, small-molecule inhibitor of EZH2 methyltransferase activity. GSK126 decrease...
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Pirodavir(R 77975)
Pirodavir(R-77975) is the prototype of a novel class of broad-spectrum antipicornavirus compounds. [1][2]
Reference:
[1] Antimicrob. Agents ...
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AMG 517
AMG-517 is a potent antagonist of TRV1. Transient receptor potential vanilloid 1 (TRPV1) channel antagonists may have clinical utility for the treatme...
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CP 809101
CP-809101 hydrochloride is a potent and selective SR-2C agonist. CP809101 displays antipsychotic activity by suppressing condition avoidance respondin...
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MLN 120B
MLN-120B is a novel IKappaB kinase (IKK)beta inhibitor. MLN120B induces growth inhibition of multiple myeloma cells in SCID-hu mouse model. [1][2]
&n...
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Clobenpropit (VUF 9153)
Clobenpropit (VUF-9153) has been shown to be an extremely potent (pA2 = 9.93) and selective histamine H3 receptor antagonist. This compound has been f...
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Nucleozin
Nucleozin targets influenza A nucleoprotein (NP), a multifunctional, RNA-binding protein necessary for virus replication. Nucleozin is effective in fi...
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KY 0211
KY-0211 promotes differentiation of human ESCs and iPSCs into cardiomyocytes. KY0211 induces downregulation of Wnt signaling target genes adn inhibits...
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MK3697
MK-3697 is an isonicotinamide small molecule, acting as a potent and selective Orexin receptor antagonist with Ki = 0.95 nM.
Chemical ...
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AG 13958
Chemical Information
Molecular Weight (WM):
467.49
...
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Revaprazan
Revaprazan (YH-1885, SB-641257) is a novel proton pump inhibitor. [1][2]
Reference:
[1] J Clin. Pharmacol. 2004, 44, 73-82..
[2] Drug ...
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Bazedoxifene
Bazedoxifene is a selective estrogen receptor modulator (SERM) currently in development for osteoporosis prevention and treatment. Preclinical and cli...
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