Linezolid

Linezolid is a synthetic antibiotic used for the treatment of serious infections caused by Gram-positive bacteria that are resistant to several other ...

More>>

LY 573636 (Tasisulam)

LY573636 (Tasisulam) activates, through an as of yet not fully elucidated mechanism, the intrinsic mitochondrial-mediated cell death pathway as manife...

More>>

(+) Etomoxir sodium salt

(+) Etomoxir sodium salt is an inhibitor of carnitine palmitoyltransferase I (CPT1). (+) Etomoxir sodium salt inhibits β-oxidation in mitochondri...

More>>

SC 26196

SC-26196 is a selective Δ6 desaturase inhibitor (IC50 = 0.2 μM in vitro). SC26196 displays selectivity over Δ5 and Δ9 desaturases...

More>>

Gadobutrol (Gadavist)

Gadobutrol (Gadavist) is a gadolinium-based MRI contrast agent (GBCA). [1] Reference: [1]Invest. Radiol. 2011, 46, 663-671. ...

More>>

Nitisinone (SC 0735)

Nitisinone (SC-0735) reversibile inhibits 4-hydroxyphenylpyruvate oxidase, thus preventing the formation of maleylacetoacetic acid and fumarylacetoace...

More>>

DCG 04

DCG-04, a biotinylated, mechanism-based probe that covalently targets mammalian cysteine proteases of the papain family was found to detect Drosophila...

More>>

Ki 16425

Ki16425 is a competitive, potent and reversible antagonist to lysophosphatidic acid (LPA1), LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 &m...

More>>

Zafirlukast

Zafirlukast is an oral leukotriene receptor antagonist (LTRA) for the maintenance treatment of asthma, often used in conjunction with an inhaled stero...

More>>

Montelukast sodium

Montelukast (MK-0476) is a leukotriene receptor antagonist (LTRA) used for the maintenance treatment of asthma and to relieve symptoms of seasonal all...

More>>

BIBR 1048 (Dabigatran, Pradaxa)

BIBR-1048 (Dabigatran, Pradaxa) is an anticoagulant from the class of the direct thrombin inhibitors. It is being studied for various clinical indicat...

More>>

Decitabine

Decitabine (Dacogen) is a potent inhibitor of DNA methylation with IC50 of 438 nM and 4.38 nM in HL-60 and KG1a cells, respectively. Decitabine is ind...

More>>

Febuxostat

Febuxostat (Uloric, Adenuric) is a non-purine selective inhibitor of xanthine oxidase. It works by non-competitively blocking the molybdenum pterin ce...

More>>

Aprepitant (MK 0869)

Aprepitant (MK-0869) is classified as an NK1 antagonist. Aprepitant (MK0869) has been shown to inhibit both the acute and delayed emesis induced by cy...

More>>

Oseltamivir (Tamiflu)

Oseltamivir (Tamiflu) is a neuraminidase inhibitor, serving as a competitive inhibitor of the activity of the viral neuraminidase (NA) enzyme upon sia...

More>>

T 705

T-705 (Favipiravir), a substituted pyrazine compound, has been found to exhibit potent anti-influenza virus activity in vitro and in vivo. In a time-o...

More>>

Total: 192 Page: 9 / 12 First ←Previous Next→ End