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Products > GPCR > Adenosine Receptor > Istradefylline (KW 6002)
Product name : Istradefylline (KW 6002)
Item : cc324
Price : 200mg, $459;500mg, $850; 1g $1195; 2g, $1795
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 155270-99-8
Molecular Weight : 384.43
Formula : C₂₀H₂₄N₄O₄
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
Istradefylline (KW-6002) is a selective adenosine A2A receptor (A2AR) antagonist with Ki of 2.2 nM.The novel adenosine A2A receptor antagonist KW-6002 has been examined for antiparkinsonian activity in MPTP-treated primates. Oral administration of KW6002 reversed motor disability in MPTP-treated common marmosets in a dose-dependent manner.  [1][2]
 
Reference:
[1] J Neurosci. 2001, 21, RC143.
[2] Exp. Neurol. 2000, 162, 321-327.
 
 
Chemical Information
Molecular Weight (WM):
384.43
Formula:
C20H24N4O4
CAS No:
155270-99-8, 861889-00-1 (6H2O), 861889-02-3 (5H2O)
Purity:
≥ 98%
Synonyms:
KW 6002
 
DMSO ≥ 6 mg/mL
Solubility (25℃)
Water < 1 mg/mL
 
Ethanol < 1 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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