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Product name : Roflumilast
Item : cc305
Price : 1g, $650;2g, $1050; 5g $1650
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 162401-32-3
Molecular Weight : 403.21
Formula : C₁₇H₁₄Cl₂F₂N₂O₃
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
Roflumilast (Daxas, Daliresp) is a drug which acts as a selective, long-acting inhibitor of the enzyme PDE-4 with an IC50 of 0.8 nM. It has antiinflammatory effects and is under development as an orally administered drug for the treatment of inflammatory conditions of the lungs such as asthma, and chronic obstructive pulmonary disease (COPD).   [1][2]
 
Reference:
[1] Int. J Chron. Obstruct. Pulmon. Dis. 2007, 2, 121-129.
[2] Clin. Exp. Allergy 2008, 38, 847-856.
 
 
Chemical Information
Molecular Weight (WM):
403.21
Formula:
C17H14Cl2F2N2O3
CAS No:
162401-32-3
Purity:
≥ 98%
Synonyms:
Daxas
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.
 

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