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A 803467
A-803467 is a selective NaV1.8 channel blocker with IC50 of 8 nM. A 803467 potently blocks recombinant human or rat NaV1.8 channels with IC50 of 8 nM ...
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Retigabine (Ezogabine)
Retigabine (Ezogabine, D-23129, Potiga, Trobalt) is an anticonvulsant for KCNQ2/3 currents with EC50 of 3.6 μM. Retigabine is a potent KCNQ channel...
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Vernakalant (RSD 1235)
Vernakalant (RSD 1235) blocks atrial potassium channels, thereby prolonging repolarization. It differs from typical class III agents by blocking a cer...
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Dronedarone (Multaq)
Dronedarone (Multaq)has been termed a “multichannel blocker” however it is unclear which channel(s) play a pivotal role in its success. Th...
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