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Product name : MPC 3100
Item : cc244
Price : 200mg, $1250;500mg, $2090; 1g $2995; 2g, $4395
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 958025-66-6
Molecular Weight : 549.4407
Formula : C22H25BrN6O4S
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
MPC-3100 is a fully synthetic potent small-molecule Hsp90 inhibitor with IC50 of 60 nM. Hsp90 inhibitor MPC3100 selectively binds to Hsp90, thereby inhibiting its chaperone function and promoting the degradation of oncogenic signaling proteins involved in tumor cell proliferation and survival; this agent may inhibit the growth and survival of a wide variety of cancer cell types. Hsp90, a chaperone protein upregulated in a variety of tumor cells, regulates the folding, stability, and degradation of many oncogenic signaling proteins. [1]
 
Reference:
[1] PCT Int. Appl. (2011), WO 2011060253 A2 20110519.
[2] PCT Int. Appl. (2007), WO 2007134298 A2 20071122.
 
 
Chemical Information
Molecular Weight (WM):
549.44
Formula:
C22H25BrN6O4S
CAS No:
958025-66-6
Purity:
≥ 98%
Synonyms:
MPC 3100
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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