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ITD-1
Description of:ITD-1
ITD-1(cas:1099644-42-4) is a selective inhibitor of TGF-β signaling (IC50 = 0.85 μM); displays little or no inhibi...
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K 02288
Chemical Information
Download K02288 SDF
Molecular Weight (MW)
352.38
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Go 6983
Go-6983 is a pan PKC inhibitor against PKCα, PKCβ, PKCγ, PKCδ, PKCζ with IC50 of 7 nM, 7 nM, 6 nM, 10 nM and 60 nM, respec...
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Bryostatin 1
Bryostatin 1 is a macrolactone isolated from the marine bryozoan, Bugula neritina, that modulates protein kinase C (PKC) activity with Ki of 1.35 nM. ...
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Staurosporine (AM 2282)
Staurosporine (AM-2282) is a potent PKC inhibitor with IC50 of 2.7 nM. It induces PKC translocation, induces association of purified PKC with inside-o...
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LY 364947
LY364947 is a potent, selective ATP-competitive inhibitor of TGFβR-I with IC50 of 59 nM. Transforming growth factor-β signals through a cell...
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CX 4945 (silmitasertib)
CX 4945 (Silmitasertib) is an orally bioavailable small-molecule inhibitor of CK2 with potential antineoplastic activity. CX-4945 selectively binds to...
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Enzastaurin (LY 317615)
Enzastaurin (LY-317615) is a potent PKC beta inhibitor for PKCβ, PKCα, PKCγ and PKCε with IC50 of 6 nM, 39 nM, 83 nM and 110 ...
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LY2109761
LY2109761 is a novel selective TGFβ receptor type I and type II (TβRI/II) dual inhibitor with Ki of 38 nM and 300 nM, respectively. Blocking...
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LY 2157299
LY2157299 is a potent TβRI and TβRII (transforming growth factor β receptor I and II) inhibitor with IC50 of 86 nM and 2 nM, respective...
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