PI 103

PI 103 is an inhibitor of DNA-PK, PI 3-kinase (p110α) and mTOR (IC50 values are 2, 8, 20, 26, 48, 83, 88, 150, 850, 920, ~ 1000 and 2300 nM for ...

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GSK 2126458

GSK 2126458 is a highly potent PI3K and mTOR inhibitor with an app Ki of 19 pM for PI3K. GSK 2126458 binds to and inhibits PI3K in the PI3K/mTOR signa...

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TGX 221

TGX 221 is a cell-permeable morpholino-pyrimidinone compound that acts as a reversible, ATP-competitive, selective, and highly potent inhibitor of PI ...

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IC 87114

IC 87114 is a cell permeable, selective inhibitor of PI 3-Kδ (IC50= 1.82, 0.07, and 1.24 for p110b, p110d, and p110g, respectively, but may also...

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AS 605240

AS 605204 is a potent and selective inhibitor of PI 3-kinase γ (PI 3-Kγ) (IC50 = 8 nM). It displays 30-fold selectivity over PI 3-Kδ...

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TG100-115

TG100-115, inhibited PI3K γ and -δ(IC50 values of 83 and 235 nM, respectively), whereas both PI3Kα and -β were relatively unaff...

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PIK 93

PIK-93 is a PI4KIIIβ inhibitor (IC50 at 19 nM). PIK-93 is the first reported PI4-kinase inhibitor, which is able to inhibit PI4KIIIβ at low-...

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LY 294002 (NSC 697286, SF 1101)

LY 294002 is a potent inhibitor of phosphoinositide 3-kinases (PI3Ks). Two of these are the proto-oncogene serine/threonine-protein kinase (PIM1) and ...

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YM 201636

YM 201636 is an inhibitor of retroviral budding and PIKfyve-catalyzed PtdIns(3,5)P2 synthesis, can halt glucose entry by insulin in adipocytes. Y...

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