Go 6976

Go-6976 is a potent protein kinase C (PKC) inhibitor (IC50 = 7.9 nM). Go6976 discriminates between Ca2+-dependent and -independent isoforms of PKC in ...

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CID 2011756

CID-2011756 is a protein kinase D (PKD) inhibitor (IC50 values are 0.6, 0.7 and 3.2 μM for PKD2, PKD3 and PKD1 respectively). Protein kinase D (PKD...

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CID 1067700

CID-1067700 is an inhibitor of nucleotide binding by Ras-related GTPases. CID1067700 has significant inhibitory potency on Rab7 nucleotide binding wit...

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CHR-6494

CHR-6494 is a first-in-class Haspin inhibitor with a wide spectrum of anticancer effects. Haspin is a serine/threonine kinase that phosphorylates Thr-...

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Pentostatin

Pentostatin is an extremely potent (Ki = 2.5 pM) irreversible inhibitor of adenosine deaminase. Pentostatin inhibition of ADA appears to result in ele...

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NSC 23766

NSC 23766 is a specific inhibitor of the binding and activation of RAC GTPase.NSC-23766Prevents Rac1 activation by Rac-specific guanine nucleotide exc...

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Minocycline

Minocycline is a broad-spectrum tetracycline antibiotic. [1][2] Reference: [1] Toxicol. Appl. Pharmacol. 1967, 11, 128-149. [2] Antim...

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Netobimin

Netobimin is an anthelmintic drug. Chemical Information Molecular Weight (WM): ...

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Tirofiban (Aggrastat)

Tirofiban (Aggrastat) is an antiplatelet drug. It belongs to a class of antiplatelet named glycoprotein IIb/IIIa inhibitors. Tirofiban is the first dr...

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OC 000459

OC000459, is a potent, selective, and orally active D prostanoid receptor 2 antagonist that inhibits mast cell-dependent activation of T helper 2 lymp...

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WZ 811

WZ811 is a C-X-C chemokine receptor type 4 (CXCR4) antagonist. WZ-811 shows subnanomolar potency (EC50 = 0.3 nM) in an affinity binding assay. The CXC...

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UNC 0638

UNC-0638 is an inhibitor of G9a and GLP with excellent potency (IC50 < 20nM) and selectivity over a wide range of epigenetic and non-epigenetic tar...

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CCG 50014

CCG-50014, the most potent small molecule RGS inhibitor to date has an IC(50) for RGS4 of 30 nM and is >20-fold selective for RGS4 over other RGS p...

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Duloxetine

Duloxetine is a serotonin-norepinephrine reuptake inhibitor (SNRI). It is effective for major depressive disorder and generalized anxiety disorder (GA...

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Peramivir (RWJ 270201, BCX1812)

Peramivir (RWJ-270201, BCX-1812) is a transition-state analogue and a potent, specific influenza viral neuraminidase inhibitor with an IC50 of median ...

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Bexarotene

Bexarotene is a retinoid specifically selective for retinoid X receptors, as opposed to the retinoic acid receptors. RXRs are located primarily in vis...

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